Teaching Plan

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TEACHING PLAN: 11NT310 – 12CH316 ADVANCED PHARMACEUTICAL CHEMISTRY Credits 4:0:0
November2012 to April 2012

Name of the Faculty member: Mr. G. Yowan Nerthigan Designation: Assistant Professor Specialization – MSc Chemistry(II year)Dept / School: Science and Humanities / School of Nanoscience and Technology Unit

No.
Lecture
No.
Topic
Book & Page Nos.
Used for teaching
Topic No.
Date Taught
Unit 1
BASICS OF MEDICINAL CHEMISTRY
1,2
Introduction to drug design
Medicinal Chemistry by Ashutosh Kar
1

3
Physical and
chemical factors associated with biological activities
Medicinal Chemistry by Ashutosh Kar
2

4,5
Classification of drugs based on structure
or pharmacological basis with examples
Medicinal Chemistry by Ashutosh Kar
3

6,7
Pro drugs and soft drugs

4

8,9
Design of pro drug system
– Multiple pro drug formation
Medicinal Chemistry by Ashutosh Kar
5

10, 11
Soft drug principle and applications
Journal Article
6

12
Quantitative Structure
Activity Relationship –
Medicinal Chemistry by Ashutosh Kar & Medicinal Chemistry by Gareth Thomas 7

13, 14
Chirality in Drug Design.
Journal Article
8

Unit II
DRUG DISCOVERY AT THE ENZYME LEVEL
15
Unit II
DRUG DISCOVERY AT THE ENZYME LEVEL

16
Enzymes and enzyme inhibitors
Medicinal Chemistry by Gareth Thomas
9

17
Competitive and non-competitive inhibitors
Medicinal Chemistry by Gareth Thomas
10

18, 19
Reversible and irreversible inhibitor
Medicinal Chemistry by Gareth Thomas
11

20, 21
Ligand receptor theories
Medicinal Chemistry by Gareth Thomas
12

22, 23
Clark’s theory and Paton’s rate theory
Medicinal Chemistry by Gareth Thomas
13

24, 25
Proteins, lipids, and nucleic acids as
drug targets
Medicinal Chemistry by Gareth Thomas
14

26, 27
Effect of pH, pKa, and polarity on drug solubility
Medicinal Chemistry by Gareth Thomas
15...
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