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Teaching Plan

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TEACHING PLAN: 11NT310 – 12CH316 ADVANCED PHARMACEUTICAL CHEMISTRY Credits 4:0:0
November2012 to April 2012

Name of the Faculty member: Mr. G. Yowan Nerthigan Designation: Assistant Professor Specialization – MSc Chemistry(II year)Dept / School: Science and Humanities / School of Nanoscience and Technology Unit

No.
Lecture
No.
Topic
Book & Page Nos.
Used for teaching
Topic No.
Date Taught
Unit 1
BASICS OF MEDICINAL CHEMISTRY
1,2
Introduction to drug design
Medicinal Chemistry by Ashutosh Kar
1

3
Physical and
chemical factors associated with biological activities
Medicinal Chemistry by Ashutosh Kar
2

4,5
Classification of drugs based on structure
or pharmacological basis with examples
Medicinal Chemistry by Ashutosh Kar
3

6,7
Pro drugs and soft drugs

4

8,9
Design of pro drug system
– Multiple pro drug formation
Medicinal Chemistry by Ashutosh Kar
5

10, 11
Soft drug principle and applications
Journal Article
6

12
Quantitative Structure
Activity Relationship –
Medicinal Chemistry by Ashutosh Kar & Medicinal Chemistry by Gareth Thomas 7

13, 14
Chirality in Drug Design.
Journal Article
8

Unit II
DRUG DISCOVERY AT THE ENZYME LEVEL
15
Unit II
DRUG DISCOVERY AT THE ENZYME LEVEL

16
Enzymes and enzyme inhibitors
Medicinal Chemistry by Gareth Thomas
9

17
Competitive and non-competitive inhibitors
Medicinal Chemistry by Gareth Thomas
10

18, 19
Reversible and irreversible inhibitor
Medicinal Chemistry by Gareth Thomas
11

20, 21
Ligand receptor theories
Medicinal Chemistry by Gareth Thomas
12

22, 23
Clark’s theory and Paton’s rate theory
Medicinal Chemistry by Gareth Thomas
13

24, 25
Proteins, lipids, and nucleic acids as
drug targets
Medicinal Chemistry by Gareth Thomas
14

26, 27
Effect of pH, pKa, and polarity on drug solubility
Medicinal Chemistry by Gareth Thomas
15...
TEACHING PLAN: 11NT310 – 12CH316 ADVANCED PHARMACEUTICAL CHEMISTRY
Credits 4:0:0
November2012 to April 2012
Name of the Faculty member: Mr. G. Yowan Nerthigan Designation: Assistant Professor
Specialization – MSc Chemistry(II year) Dept / School: Science and Humanities /
School of Nanoscience and Technology
Unit
No.
Lecture
No. Topic Book & Page Nos.
Used for teaching Topic No. Date
Taught
Unit 1
BASICS OF MEDICINAL CHEMISTRY
1,2 Introduction to drug design Medicinal Chemistry by Ashutosh
Kar 1
3
Physical and
chemical factors associated with
biological activities
Medicinal Chemistry by Ashutosh
Kar 2
4,5
Classification of drugs based on
structure
or pharmacological basis with
examples
Medicinal Chemistry by Ashutosh
Kar 3
6,7 Pro drugs and soft drugs 4
8,9 Design of pro drug system
– Multiple pro drug formation
Medicinal Chemistry by Ashutosh
Kar 5
10, 11 Soft drug principle and applications Journal Article 6
12 Quantitative Structure
Activity Relationship –
Medicinal Chemistry by Ashutosh
Kar & Medicinal Chemistry by
Gareth Thomas
7
13, 14 Chirality in Drug Design. Journal Article 8
Unit II
15
Unit II
DRUG DISCOVERY AT THE
ENZYME LEVEL
16 Enzymes and enzyme inhibitors Medicinal Chemistry by Gareth
Thomas 9
17 Competitive and non-competitive
inhibitors
Medicinal Chemistry by Gareth
Thomas 10
18, 19 Reversible and irreversible inhibitor Medicinal Chemistry by Gareth
Thomas 11
20, 21 Ligand receptor theories Medicinal Chemistry by Gareth
Thomas 12
22, 23 Clark’s theory and Paton’s rate theory Medicinal Chemistry by Gareth
Thomas 13
24, 25 Proteins, lipids, and nucleic acids as
drug targets
Medicinal Chemistry by Gareth
Thomas 14
26, 27 Effect of pH, pKa, and polarity on
drug solubility
Medicinal Chemistry by Gareth
Thomas 15
28 DNA Protein interaction and Medicinal Chemistry by Ashutosh 16